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Transformation of substituted 3-hydroxy-4-[(2E)-3-arylprop-2-enoyl]-1,5-dihydro-2H-pyrrol-2-ones by the action of I2/DMSO into derivatives 2-aryl-5,6-dihydropyrano[2,3-c]pyrrole-4,7-diones

JOURNAL ARTICLE published 30 December 2021 in Ukrainica Bioorganica Acta

Authors: Roman Vydzhak | Svitlana Panchishin | Yaroslav Prostota | Volodymyr Brovarets

Chemistry of difluoromethylene phosphonates: history, state of the art, and prospects

JOURNAL ARTICLE published 30 June 2022 in Ukr. Bioorg. Acta 2022, Vol. 17, N1

Research funded by Bundesministerium für Wirtschaft und Energie (“GO3” project No. 03ETE002C)

Authors: Mykhailo Shevchuk | Gerd-Volker Röschenthaler

Aldol Addition-Cyclization Reaction Cascade on a Platform of Chiral Ni(II) Complex of Glycine Schiff Base

JOURNAL ARTICLE published 30 June 2021 in Ukr. Bioorg. Acta 2021, Vol. 16, N1

Research funded by Foundation for Innovative Research Groups of the National Natural Science Foundation of China (21761132021)

Authors: Yupiao Zou | Zizhen Yin | Haibo Mei | Hiroyuki Konno | Hiroki Moriwaki | Vadim Soloshonok | Jianlin Han

Anticancer evaluation of di- and trifunctional substituted 1,3-thiazoles

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Kostyantyn Turov | Оleg Mitiukhin | Svitlana Chumachenko | Vladimir Zyabrev | Volodymyr Brovarets

In vitro and in silico study of 1,3-oxazol-4-yltriphenylphosphonium salts as potential inhibitors of Candida albicans transglycosylase

JOURNAL ARTICLE published 30 June 2021 in Ukr. Bioorg. Acta 2021, Vol. 16, N1

Research funded by National Research Foundation of Ukraine (2020.01/0075)

Authors: Ivan Semenyuta | Maria Trush | Diana Hodyna | Maryna Kachaeva | Larysa Metelytsia | Volodymyr Brovarets

Theoretical evaluation of electroanalitical determination of diazoline (mebhydrolin) on a polymer electrode

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Volodymyr Tkach | Marta Kushnir | Yana Ivanushko | Silvio de Oliveira | Olga Luganska | Petro Yagodynets | Zholt Kormosh

The main directions of scientific activity of Academician V.P. Kukhar

JOURNAL ARTICLE published 30 June 2022 in Ukr. Bioorg. Acta 2022, Vol. 17, N1

Research funded by National Academy of Sciences of Ukraine (01190100611)

Authors: Vadim Romanenko

Cytisine derivatives as new anti-Escherichia coli agents: in silico and in vitro studies

JOURNAL ARTICLE published 30 December 2021 in Ukrainica Bioorganica Acta

Authors: Diana Hodyna | Vasyl Kovalishyn | Volodymyr Blagodatnyi | Svitlana Bondarenko | Galyna Mrug | Mykhaylo Frasinyuk | Larysa Metelytsia

The mathematical description of dopamine electrochemical oxidation, accompanied by its chemical and electrochemical polymerization

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Volodymyr Tkach | Marta Kushnir | Yana Ivanushko | Svitlana Lukanova | Silvio C. de Oliveira | Petro Yagodynets

5-Substituted N-(9H-purin-6-yl)-1,2-oxazole-3-carboxamides as xanthine oxidase inhibitors

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Research funded by National Academy of Sciences of Ukraine (CPDF 1-17)

Authors: Oksana Muzychka | Olexandr Kobzar | Oleg Shablykin | Volodymyr Brovarets | Andriy Vovk

4-(1-Oxo-1H-isochromen-3-yl)benzenesulfonamides and their effect on cancer cell growth

JOURNAL ARTICLE published 30 December 2021 in Ukrainica Bioorganica Acta

Authors: Serhii Hlotov | Olga Shablykina | Volodymyr Khilya

Fluorinated NH-iminophosphonates in synthesis of biorelevant α-aminophosphonic acids derivatives

JOURNAL ARTICLE published 30 June 2022 in Ukr. Bioorg. Acta 2022, Vol. 17, N1

Authors: Yulia Rassukana | Ivanna Yelenich | Petro Onysʹko

In silico study of binding affinity of nitrogenous bicyclic heterocycles: fragment-to-fragment approach

JOURNAL ARTICLE published 30 December 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N2

Authors: Yevheniia Velihina | Nataliya Obernikhina | Stepan Pilyo | Maryna Kachaeva | Oleksiy Kachkovsky | Volodymyr Brovarets

Nitro-substituted aurones as xanthine oxidase inhibitors

JOURNAL ARTICLE published 30 December 2021 in Ukrainica Bioorganica Acta

Authors: Oleksandr Kobzar | Iryna Mischenko | Alona Tatarchuk | Vasyl Vdovin | Sergiy Lukashov | Sergiy Yarmoluk | Andriy Vovk

Investigation of the extract's composition of Viper's bugloss (Echium vulgare)

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Anna Kapusterynska | Vira Hamada | Anna Krvavych | Roksolana Konechna | Maria Kurka | Volodymyr Novikov

Indole alkaloid ellipticine as efficient multitarget compound

JOURNAL ARTICLE published 30 June 2022 in Ukr. Bioorg. Acta 2022, Vol. 17, N1

Research funded by Horizon 2020 (MSCA-RISE-2016-734759)

Authors: Kostiantyn Shvydenko | Iryna Grafova | Tetiana Shvydenko | Aleksandr Kostyuk | Neila Picanço | Luiz Silva | Anya Kropfitsch | Claudia Wyrepkowski | Luiz Zerbini | Wanderli Tadei | Antonia Pereira | Markku Leskelä | Andriy Grafov

Сationic carboxamide derivatives of tricyclic heteroaromatic compounds: synthesis and preliminary evaluation of antiproliferative activity

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Valentina Kostina | Inna Alexeeva | Nadia Lysenko | Valentina Negrutska | Igor Dubey

Three-component cyclization as an approach to a combinatorial library of 2H-spiro-[chromeno[2,3-c]pyrrole-1,3'-indoline]-2',3,9-triones

JOURNAL ARTICLE published 30 June 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N1

Authors: Roman Vydzhak | Maryna Kachaeva | Stepan Pilyo | Viktoriia Moskvina | Olga Shablykina | Andriy Kozytskiy | Volodymyr Brovarets

Synthesis of fluorinated pyrrolizidine, indolizidine and quinolizidine derivatives

JOURNAL ARTICLE published 30 June 2022 in Ukr. Bioorg. Acta 2022, Vol. 17, N1

Research funded by National Academy of Sciences of Ukraine (2.1.10.19-22)

Authors: Anton Klipkov | Igor Gerus | Alexander Sorochinsky

Features of the synthesis and biological evaluation of 3-(carboxyphenyl)chromones

JOURNAL ARTICLE published 30 December 2020 in Ukr. Bioorg. Acta 2020, Vol. 15, N2

Research funded by Ministry of Education and Science of Ukraine (19БФ037-03)

Authors: Olga Shablykina | Viktoriia Moskvina | Volodymyr Khilya